Skip to content
PeptideHormone

Glucose-dependent insulinotropic polypeptide vs Tirzepatide

The second incretin, with distinct adipose and CNS biology. A dual GIP and GLP-1 receptor agonist — the first of the co-agonists. Side by side: type, evidence tier, receptor, molecular weight, and half-life — the same fields as each monograph, rearranged so the engineering difference is visible.

Glucose-dependent insulinotropic polypeptide
GIP
Tirzepatide
Also known asMounjaro, Zepbound
TypeEndogenousAnalog
EvidenceEstablishedEstablished
FamilyIncretins & metabolicIncretins & metabolic
ClassIncretin peptide (42 aa)Dual GIP/GLP-1 receptor agonist (39 aa, acylated)
ReceptorGIP receptor (GIPR), a class B GPCRGIP receptor + GLP-1 receptor
Molecular weight~4,983.6 Da~4,813.5 Da
Half-life
~5–7 min (native; DPP-4)
Model dosing
~5 days (~120 h)
Model dosing
Based onNative hormoneGlucose-dependent insulinotropic polypeptide

Half-life bars are on a logarithmic scale across the molecules shown. Reference values for the native or representative form — educational only, not medical or dosing advice.

Common questions

What is the difference between Glucose-dependent insulinotropic polypeptide and Tirzepatide?
Glucose-dependent insulinotropic polypeptide is an endogenous hormone; Tirzepatide is an engineered analog based on Glucose-dependent insulinotropic polypeptide. Glucose-dependent insulinotropic polypeptide signals at GIP receptor (GIPR), a class B GPCR; Tirzepatide signals at GIP receptor + GLP-1 receptor.
How do the half-lives of GIP and Tirzepatide compare?
The reported circulating half-life of Glucose-dependent insulinotropic polypeptide is ~5–7 min (native; DPP-4); Tirzepatide is ~5 days (~120 h). These are reference values for the native or representative form — educational only, not dosing advice.

Prefer the other order? Tirzepatide vs Glucose-dependent insulinotropic polypeptide. Or open the interactive comparison tool to add more molecules.