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PeptideHormone

Retatrutide vs Brenipatide

An investigational GIP/GLP-1/glucagon triple receptor agonist. A once-monthly dual GIP/GLP-1 agonist aimed at the brain's reward circuitry rather than the scale. Side by side: type, evidence tier, receptor, molecular weight, and half-life — the same fields as each monograph, rearranged so the engineering difference is visible.

Retatrutide
Brenipatide
LY3537031
Also known as
TypeAnalogAnalog
EvidenceInvestigationalInvestigational
FamilyIncretins & metabolicIncretins & metabolic
ClassGIP/GLP-1/glucagon triple agonist (acylated peptide)GIP/GLP-1 dual agonist (acylated peptide)
ReceptorGIP + GLP-1 + glucagon receptorsGIP + GLP-1 receptors
Molecular weight4,900 Da4,900 Da
Half-lifeengineered for once-monthly dosing
Based onGlucagon-like peptide-1Glucagon-like peptide-1

Half-life bars are on a logarithmic scale across the molecules shown. Reference values for the native or representative form — educational only, not medical or dosing advice.

Common questions

What is the difference between Retatrutide and Brenipatide?
Retatrutide is an engineered analog based on Glucagon-like peptide-1; Brenipatide is an engineered analog based on Glucagon-like peptide-1. Retatrutide signals at GIP + GLP-1 + glucagon receptors; Brenipatide signals at GIP + GLP-1 receptors.
How do the half-lives of Retatrutide and LY3537031 compare?
The reported circulating half-life of Retatrutide is ~6 days; Brenipatide is engineered for once-monthly dosing. These are reference values for the native or representative form — educational only, not dosing advice.

Prefer the other order? Brenipatide vs Retatrutide. Or open the interactive comparison tool to add more molecules.